Contents
Letters in Drug Design & Discovery, Volume 13 - Number 9
Structure-based Drugs Design Studies on Spleen Tyrosine Kinase Inhibitors
, 13(9): 845 - 858Letícia Cristina Assis, Letícia Santos Garcia, Daiana Teixeira Mancini, Tamiris Maria Assis, Daniela Rodrigues Silva, Giovanna Gajo Cardoso, Alexandre Alves de Castro, Teodorico Castro Ramalho and Elaine Fontes Ferreira da Cunha.
DOI: 10.2174/1570180813666160725095118
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In-silico Designing of Novel Camptothecin Analogues as Potent Inhibitors of Topoisomerase I: A Molecular Docking, QSAR, and ADME-T Study
, 13(9): 859 - 868Darpan Raghav, Babukrishna Maniyadath, Aruna Mohan, Sutari Sairam, Rinu Mary Rajan and Krishnan Rathinasamy.
DOI: 10.2174/1570180813666160518123550
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Synthesis, Biological Evaluation and in silico Studies of Novel 5α-aza-Bhomo-3,5-secosteroids as Potential 5-reductase Inhibitors
, 13(9): 869 - 878Rajnish Kumar, Pankaj Chauhan, Priyanka Malla, Manoj K. Mahapatra, Rolf W. Hartmann, Jörg Haupenthal and Manoj Kumar.
DOI: 10.2174/1570180813666160630110649
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Identification of Novel IRAK-4 Inhibitors Through Pharmacophore Modeling, Atom-based 3D-QSAR, Docking Strategies and Molecular Dynamics Simulation
,13(9): 879 - 887Liangliang Zhong, Lu Zhou, Yahui Tian and Rong You.
DOI: 10.2174/1570180813666160421163027
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Imidazole-based Derivatives as Potential Anti-platelet Inhibitors: DFT and Molecular Docking Study
, 13(9): 888 - 896Mehbub I. K. Momin, Neil A. Koorbanally and Bahareh Honarparvar.
DOI: 10.2174/1570180813666160517162937
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Synthesis and Antiacetylcholinesterase Activity Evaluation of New 2-aryl Benzofuran Derivatives
, 13(9): 897 - 902Behjat Pouramiri, Mohammad Mahdavi, Setareh Moghimi, Loghman Firoozpour, Hamid Nadri, Alireza Moradi, Esmat Tavakolinejad-Kermani, Ali Asadipourand Alireza Foroumadi.
DOI: 10.2174/1570180813666160610124637
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Synthesis and Evaluation of New Thiazole Derivatives as Potential Antimicrobial Agents
, 13(9): 903 - 911Mehlika Dilek Altıntop, Ahmet Özdemir, Özlem Atlı, Zerrin Cantürk, Merve Baysal and Zafer Asım Kaplancıklı.
DOI: 10.2174/1570180813666160226001021
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Synthesis and In vivo Antifibrotic Activity of Novel Leflunomide Analogues
, 13(9): 912 - 920Abdelrahman Hamdi, Eman Said, Abdelbasset A. Farahat, Serry A. A. El-Bialy and Mohammed A M Massoud.
DOI: 10.2174/1570180813666160630125624
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Synthesis and Antimicrobial Evaluation of New Pyrazoline and Pyrazolinyl Thiazole Derivatives Bearing Tetrazolo[1,5-a]quinoline Moiety
, 13(9): 921 - 931Ibrahim A. M. Radini, Rizk E. Khidre and Emad M El-Telbani.
DOI: 10.2174/1570180813666160712234454
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Design, Synthesis and Antimalarial Activity of Some New Aminoalcoholpyrrolo[1,2-a]quinoxaline Derivatives
, 13(9): 932 - 942Jean Guillon, Stéphane Moreau, Luisa Ronga, Louise Basmacyian, Anita Cohen, Sandra Rubio, Guillaume Bentzinger, Solène Savrimoutou, Nadine Azas,Catherine Mullié and Pascal Sonnet.
DOI: 10.2174/1570180813666160517164758
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Significance of Amino Group Substitution at Combretastatin A-4 and Phenstatin Analogs
, 13(9): 943 - 951Vijay K. Patel and Harish Rajak.
DOI: 10.2174/1570180813666160517163444
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Study of Some Piperine Analogues on Drugs Efflux by Targeting P-glycoprotein, an in silico Approach
, 13(9): 952 - 961Anushree Tripathi, Krishna Misra and Rajesh Kumar Kesharwani.
DOI: 10.2174/1570180813999160830102312
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Sodium Channel Blocking Activity and In-vivo Testing of New Phenylimidazole Derivatives
, 13(9): 962 - 967Mirko Rivara, Manoj K. Patel, Alberto Rapalli and Valentina Zuliani.
DOI: 10.2174/1570180813666160714125755
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An Efficient Nonconventional Glycerol-Based Solid Acid Catalyzed Synthesis and Biological Evaluation of Phosphonate Conjugates of 1,2,4-triazole Thiones
,13(9): 968 - 981Madugula S. R. Murty, Mohana R. Katiki, Busam R. Rao, Sai S. Narayanan, Ruby J. Anto, Sudhreer K. Buddana, Reddy S. Prakasham, Bethala L. A. P. Devi andRachapudi B N Prasad.
DOI: 10.2174/1570180813666160125222334
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Design, Synthesis and Molecular Docking Studies of 2-Aryl/Heteroaryl-Ethyl 6-Chloroquinoline-4-Carboxylates as Potential Antimalarial Agents
, 13(9): 982 - 991Thamatakallu O. S. Kumar, Kittappa M. Mahadevan, Pasura S. Sujanganapathy and Manikyanahally N Kumara.
DOI: 10.2174/1570180813666160722112725
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